TargetMol

Denagliptin tosylate

Product Code:
 
TAR-T31378
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T31378-5mg5mg£850.00
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Quantity:
TAR-T31378-50mg50mg£1,661.00
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Quantity:
TAR-T31378-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
Denagliptin (GW823093 or GSK-823093) is a dipeptidyl peptidase IV (DPP-IV) inhibitor.
CAS:
811432-66-3
Formula:
C27H26F3N3O4S
Molecular Weight:
545.58
Purity:
0.98
SMILES:
Cc1ccc(cc1)S(O)(=O)=O.N[C@@H](C(c1ccc(F)cc1)c1ccc(F)cc1)C(=O)N1C[C@@H](F)C[C@H]1C#N

References

1. De Serres M, Bowers G, Boyle G, Beaumont C, Castellino S, Sigafoos J, Dave M, Roberts A, Shah V, Olson K, Patel D, Wagner D, Yeager R, Serabjit-Singh C. Evaluation of a chimeric (uPA+/+)/SCID mouse model with a humanized liver for prediction of human metabolism. Xenobiotica. 2011 Jun;41(6):464-75. doi: 10.3109/00498254.2011.560295. Epub 2011 Mar 4. PubMed PMID: 21370990. 2. Joshi BK, Ramsey B, Johnson B, Patterson DE, Powers J, Facchine KL, Osterhout M, Leblanc MP, Bryant-Mills R, Copley RC, Sides SL. Elucidating the pathways of degradation of denagliptin. J Pharm Sci. 2010 Jul;99(7):3030-40. doi: 10.1002/jps.22069. PubMed PMID: 20112433.