TargetMol

Dasolampanel

Product Code:
 
TAR-T31208
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T31208-5mg5mg£1,348.00
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TAR-T31208-50mg50mg£3,107.00
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TAR-T31208-100mg100mg£4,247.00
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This product comes from: United States.
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Further Information

Bioactivity:
Dasolampanel(NGX-426) is an oral bioavailable analog of tezampanel and therefore a competitive antagonist of AMPA and red alginine receptors, being developed for the treatment of chronic pain disorders, including neuropathic pain and migraine.
CAS:
503294-13-1
Formula:
C17H20ClN5O3
Molecular Weight:
377.83
Purity:
0.98
SMILES:
[H][C@@]12CC[C@@H](C[C@]1([H])C[C@H](NC2)C(O)=O)Oc1cccc(Cl)c1-c1nnn[nH]1

References

1. Wallace MS, Lam V, Schettler J. NGX426, an oral AMPA-kainate antagonist, is effective in human capsaicin-induced pain and hyperalgesia. Pain Med. 2012 Dec;13(12):1601-10. doi: 10.1111/j.1526-4637.2012.01509.x. Epub 2012 Oct 30. PubMed PMID: 23110368.