TargetMol

CGP-20712

Product Code:
 
TAR-T30846
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T30846-1mg1mg£352.00
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TAR-T30846-5mg5mg£736.00
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TAR-T30846-10mg10mg£978.00
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TAR-T30846-25mg25mg£1,348.00
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TAR-T30846-50mg50mg£1,661.00
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Quantity:
TAR-T30846-100mg100mg£2,079.00
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Quantity:
TAR-T30846-500mg500mg£4,006.00
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This product comes from: United States.
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Further Information

Bioactivity:
CGP-20712 is a beta1-selective beta-adrenoceptor antagonist.
CAS:
137888-49-4
Formula:
C23H25F3N4O5
Molecular Weight:
494.471
Pathway:
GPCR/G Protein|Neuroscience
Purity:
0.98
SMILES:
Cn1cc(nc1-c1ccc(OCC(O)CNCCOc2ccc(O)c(c2)C(N)=O)cc1)C(F)(F)F
Target:
Adrenergic Receptor

References

1. Dooley DJ, Bittiger H. Quantitative assessment of central beta 1- and beta 2-adrenoceptor regulation using CGP 20712 A. J Pharmacol Methods. 1987 Sep;18(2):131-6. PubMed PMID: 2887701. 2. Dooley DJ, Bittiger H, Reymann NC. CGP 20712 A: a useful tool for quantitating beta 1- and beta 2-adrenoceptors. Eur J Pharmacol. 1986 Oct 14;130(1-2):137-9. PubMed PMID: 2877892. 3. Kaumann AJ. The beta 1-adrenoceptor antagonist CGP 20712 A unmasks beta 2-adrenoceptors activated by (-)-adrenaline in rat sinoatrial node. Naunyn Schmiedebergs Arch Pharmacol. 1986 Apr;332(4):406-9. PubMed PMID: 2874503.