TargetMol

BMS-187308

Product Code:
 
TAR-T30498
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T30498-5mg5mg£1,171.00
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TAR-T30498-50mg50mg£2,303.00
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Quantity:
TAR-T30498-100mg100mg£3,042.00
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Further Information

Bioactivity:
BMS-187308 is an endothelin-A (ETA) selective antagonist.
CAS:
153624-15-8
Formula:
C21H25N3O3S
Molecular Weight:
399.51
Purity:
0.98
SMILES:
CC(C)Cc1ccc(c(N)c1)-c1ccccc1S(=O)(=O)Nc1onc(C)c1C

References

1. Murugesan N, Gu Z, Stein PD,et al. Biphenylsulfonamide endothelin antagonists: structure-activity relationships of a series of mono- and disubstituted analogues and pharmacology of the orally active endothelin antagonist 2'-amino-N- (3,4-dimethyl-5-isoxazolyl)-4'-(2-methylpropyl)[1, 1'-biphenyl]-2-sulfonamide (BMS-187308). J Med Chem. 1998 Dec 17;41(26):5198-218. PubMed PMID: 9857090.