TargetMol

SB-215505

Product Code:
 
TAR-T28680
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T28680-5mg5mg£850.00
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TAR-T28680-50mg50mg£1,661.00
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Quantity:
TAR-T28680-100mg100mg£2,079.00
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Further Information

Bioactivity:
SB215505 is a potent 5-HT2B/2C receptor antagonist (pKi values are 8.3, 7.66 and 6.77 for 5-HT2B, 5-HT2C and 5-HT2A respectively). It Increases wakefulness and motor activity in rats.
CAS:
162100-15-4
Formula:
C19H16ClN3O
Molecular Weight:
337.81
Purity:
0.98
SMILES:
Cc1cc2CCN(C(=O)Nc3cccc4ncccc34)c2cc1Cl

References

1. Kantor S, Jakus R, Balogh B, Benko A, Bagdy G. Increased wakefulness, motor activity and decreased theta activity after blockade of the 5-HT2B receptor by the subtype-selective antagonist SB-215505. Br J Pharmacol. 2004 Aug;142(8):1332-42. Epub 2004 Jul 20. PubMed PMID: 15265808; PubMed Central PMCID: PMC1575194.