TargetMol

RU5135

Product Code:
 
TAR-T28624
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T28624-5mg5mg£2,054.00
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Quantity:
TAR-T28624-50mg50mg£4,070.00
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Quantity:
TAR-T28624-100mg100mg£5,693.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
RU5135 is a novel convulsant amidine steroid which inhibits gamma-aminobutyric acid receptor binding.
CAS:
78774-26-2
Formula:
C18H28N2O2
Molecular Weight:
304.434
Purity:
0.98
SMILES:
[H][C@@]12CC(N)=N[C@@]1(C)CC(=O)[C@@]1([H])[C@@]2([H])CC[C@]2([H])C[C@@H](O)CC[C@]12C

References

1. Simmonds MA, Turner JP. Antagonism of inhibitory amino acids by the steroid derivative RU5135. Br J Pharmacol. 1985 Mar;84(3):631-5. PubMed PMID: 3986429; PubMed Central PMCID: PMC1987146. 2. Olsen RW. gamma-Aminobutyric acid receptor binding antagonism by the amidine steroid RU5135. Eur J Pharmacol. 1984 Aug 17;103(3-4):333-7. PubMed PMID: 6092106.