TargetMol

Profadol hydrochloride

Product Code:
 
TAR-T28452
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T28452-5mg5mg£850.00
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TAR-T28452-50mg50mg£1,661.00
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Quantity:
TAR-T28452-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
Profadol hydrochloride acts as a mixed agonist-antagonist of the μ-opioid receptor with analgesic activity.
CAS:
2324-94-9
Formula:
C14H22ClNO
Molecular Weight:
255.79
Purity:
0.98
SMILES:
Cl.CCCC1(CCN(C)C1)c1cccc(O)c1

References

1. Picker MJ, Smith MA, Morgan D. Assessment of the relative intrinsic efficacy of profadol and meperidine in a pigeon drug discrimination procedure: relevance to partial substitution patterns. Behav Pharmacol. 1994 Feb;5(1):61-70. PubMed PMID: 11224252. 2. Rhodes KF. Yohimbine antagonism of the inhibitory effects of pethidine and profadol in the mouse isolated vas deferens. J Pharm Pharmacol. 1983 Mar;35(3):182-3. PubMed PMID: 6132980. 3. Crooks PA, Sommerville R. The synthesis and analgesic activities of some spiro[indan-1,3'-pyrrolidine] derivatives designed as rigid analogs of profadol. J Pharm Sci. 1982 Mar;71(3):291-4. PubMed PMID: 6461753. 4. Leander JD. Effects of profadol on operant behavior in the pigeon. Pharmacol Biochem Behav. 1982 Mar;16(3):487-90. PubMed PMID: 6210915.