TargetMol

PD 132002

Product Code:
 
TAR-T28328
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T28328-5mg5mg£1,251.00
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TAR-T28328-50mg50mg£2,464.00
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Quantity:
TAR-T28328-100mg100mg£3,283.00
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This product comes from: United States.
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Further Information

Bioactivity:
PD 132002 is a renin inhibitor.
CAS:
134452-04-3
Formula:
C31H50N4O9S
Molecular Weight:
654.82
Purity:
0.98
SMILES:
COC(=O)[C@H](N([C@@H](CC1CCCCC1)C(O)[C@@H](O)CC(C)C)C(=O)[C@H](Cc1ccccc1)NS(=O)(=O)N1CCOCC1)C(N)=O

References

1. Palmer RK, Rapundalo ST, Batley BL, Barnes AE, Singh S, Ryan MJ, Taylor DG Jr. Disparity between blood pressure and PRA inhibition after administration of a renin inhibitor to anesthetized dogs: methodological considerations. Clin Exp Hypertens. 1993 Jul;15(4):663-81. PubMed PMID: 8374609. 2. Repine JT, Himmelsbach RJ, Hodges JC, Kaltenbronn JS, Sircar I, Skeean RW, Brennan ST, Hurley TR, Lunney E, Humblet CC, et al. Renin inhibitors containing esters at the P2-position. Oral activity in a derivative of methyl aminomalonate. J Med Chem. 1991 Jul;34(7):1935-43. PubMed PMID: 2066966.