TargetMol

OMDM169

Product Code:
 
TAR-T28235
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T28235-5mg5mg£1,492.00
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TAR-T28235-50mg50mg£2,946.00
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Quantity:
TAR-T28235-100mg100mg£4,006.00
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This product comes from: United States.
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Further Information

Bioactivity:
OMDM169 is a potent and selective MAGL inhibitor. OMDM169 could enhances 2-AG levels and of exerts analgesic activity via indirect activation of cannabinoid receptors. OMDM169 exhibited 0.13 microM10 microM).
CAS:
130193-44-1
Formula:
C25H45NO5
Molecular Weight:
439.637
Purity:
0.98
SMILES:
CCCCCCCCCCC[C@@H](C[C@@H]1OC(=O)[C@H]1CCCCCC)OC(=O)CNC=O

References

1. Valdeolivas S, Pazos MR, Bisogno T, Piscitelli F, Iannotti FA, Allar? M, Sagredo O, Di Marzo V, Fern?ndez-Ruiz J. The inhibition of 2-arachidonoyl-glycerol (2-AG) biosynthesis, rather than enhancing striatal damage, protects striatal neurons from malonate-induced death: a potential role of cyclooxygenase-2-dependent metabolism of 2-AG. Cell Death Dis. 2013 Oct 17;4:e862. doi: 10.1038/cddis.2013.387. PubMed PMID: 24136226; PubMed Central PMCID: PMC3920947. 2. Bisogno T, Ortar G, Petrosino S, Morera E, Palazzo E, Nalli M, Maione S, Di Marzo V; Endocannabinoid Research Group. Development of a potent inhibitor of 2-arachidonoylglycerol hydrolysis with antinociceptive activity in vivo. Biochim Biophys Acta. 2009 Jan;1791(1):53-60. doi: 10.1016/j.bbalip.2008.10.007. Epub 2008 Nov 5. PubMed PMID: 19027877.