TargetMol

LY 164929

Product Code:
 
TAR-T27878
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27878-5mg5mg£850.00
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TAR-T27878-50mg50mg£1,661.00
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Quantity:
TAR-T27878-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
LY 164929 is a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding site.
CAS:
113573-18-5
Formula:
C28H41N5O4
Molecular Weight:
511.667
Purity:
0.98
SMILES:
CCN(CC(=O)NC(=O)[C@@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC)[C@H](CN(C)C)Cc1ccccc1

References

1. Kim CH, Rothman RB, Jacobson AE, Mattson MV, Bykov V, Streaty RA, Klee WA, George C, Long JB, Rice KC. Probes for narcotic receptor mediated phenomena. 15. (3S,4S)-(+)-trans-3-methylfentanyl isothiocyanate, a potent site-directed acylating agent for the delta opioid receptors in vitro. J Med Chem. 1989 Jun;32(6):1392-8. PubMed PMID: 2542560. 2. Rothman RB, Long JB, Bykov V, Jacobson AE, Rice KC, Holaday JW. beta-FNA binds irreversibly to the opiate receptor complex: in vivo and in vitro evidence. J Pharmacol Exp Ther. 1988 Nov;247(2):405-16. PubMed PMID: 2846819. 3. Rothman RB, Bykov V, Ofri D, Rice KC. LY164929: a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding site. Neuropeptides. 1988 Jan;11(1):13-6. PubMed PMID: 2835701.