TargetMol

Itriglumide

Product Code:
 
TAR-T27640
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27640-5mg5mg£850.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T27640-50mg50mg£1,661.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T27640-100mg100mg£2,079.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Itriglumide, a CCK2 receptor antagonist, is used potentially for the treatment of peptic ulcers, dyspepsia, and gastroesophageal reflux disease (GERD).
CAS:
201605-51-8
Formula:
C33H38N2O4
Molecular Weight:
526.677
Purity:
0.98
SMILES:
Cc1cc(C)c(NC(=O)C[C@H](CC(O)=O)c2cccc3ccccc23)c(c1)C(=O)N1CCC2(CCCC2)CC1

References

1. Ekstr?m J, Cevik Aras H. Parasympathetic non-adrenergic, non-cholinergic transmission in rat parotid glands: effects of cholecystokinin-A and -B receptor antagonists on the secretory response. Regul Pept. 2008 Feb 7;146(1-3):278-84. Epub 2007 Oct 22. PubMed PMID: 18006087. 2. Danzer M, Jocic M, Samberger C, Painsipp E, Bock E, Pabst MA, Crailsheim K, Schicho R, Lippe IT, Holzer P. Stomach-brain communication by vagal afferents in response to luminal acid backdiffusion, gastrin, and gastric acid secretion. Am J Physiol Gastrointest Liver Physiol. 2004 Mar;286(3):G403-11. Epub 2003 Oct 30. PubMed PMID: 14592947. 3. Cevik Aras H, Ekstr?m J. Pentagastrin-induced protein synthesis in the parotid gland of the anaesthetized rat, and its dependence on CCK-A and -B receptors and nitric oxide generation. Exp Physiol. 2006 Jul;91(4):673-9. Epub 2006 Mar 23. PubMed PMID: 16556659. 4. Aras HC, Ekstr?m J. Cholecystokinin- and gastrin-induced protein and amylase secretion from the parotid gland of the anaesthetized rat. Regul Pept. 2006 May 15;134(2-3):89-96. Epub 2006 Mar 2. PubMed PMID: 16515811.