TargetMol

GIC1001 CTB salt

Product Code:
 
TAR-T27413
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27413-5mg5mg£850.00
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TAR-T27413-50mg50mg£1,661.00
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Quantity:
TAR-T27413-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
GIC-1001 is an opioid receptor agonist.
CAS:
1456509-46-8
Formula:
C29H36N2O8S2
Molecular Weight:
604.73
Purity:
0.98
SMILES:
NC(=S)c1cccc(c1)S(O)(=O)=O.CCC(COC(=O)c1cc(OC)c(OC)c(OC)c1)(N(C)C)c1ccccc1

References

1. Paquette JM, Rufiange M, Iovu Niculita M, Massicotte J, Lefebvre M, Colin P, Telmat A, Ranger M. Safety, tolerability and pharmacokinetics of trimebutine 3-thiocarbamoylbenzenesulfonate (GIC-1001) in a randomized phase I integrated design study: single and multiple ascending doses and effect of food in healthy volunteers. Clin Ther. 2014 Nov 1;36(11):1650-64. doi: 10.1016/j.clinthera.2014.08.005. PubMed PMID: 25224876. 2. Cenac N, Castro M, Desormeaux C, Colin P, Sie M, Ranger M, Vergnolle N. A novel orally administered trimebutine compound (GIC-1001) is anti-nociceptive and features peripheral opioid agonistic activity and Hydrogen Sulphide-releasing capacity in mice. Eur J Pain. 2016 May;20(5):723-30. doi: 10.1002/ejp.798. PubMed PMID: 26541237. 3. Montpetit H, Ranger M, Colin P, Furtado M, Garofolo F. Discovery of a novel trimebutine metabolite and its impact on N-desmethyltrimebutine quantification by LC-MS/MS. Bioanalysis. 2015;7(8):1007-15. doi: 10.4155/bio.15.31. PubMed PMID: 25966011.