TargetMol

Deramciclane fumarate

Product Code:
 
TAR-T27149
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27149-5mg5mg£850.00
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TAR-T27149-50mg50mg£1,661.00
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Quantity:
TAR-T27149-100mg100mg£2,079.00
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Further Information

Bioactivity:
Deramciclane fumarate is a 5-HT(2A/C) antagonist with putative anxiolytic activity.
CAS:
120444-72-6
Formula:
C24H35NO5
Molecular Weight:
417.546
Purity:
0.98
SMILES:
OC(=O)C=CC(O)=O.[H][C@]12CC[C@](C)(C1(C)C)[C@@](C2)(OCCN(C)C)c1ccccc1

References

1. K??ri?inen TM, Lehtonen M, Forsberg MM, Savolainen J, K?enm?ki M, M?nnist? PT. Comparison of the effects of deramciclane, ritanserin and buspirone on extracellular dopamine and its metabolites in striatum and nucleus accumbens of freely moving rats. Basic Clin Pharmacol Toxicol. 2008 Jan;102(1):50-8. Epub 2007 Oct 25. PubMed PMID: 17971064. 2. Al-Behaisi S, Antal I, Morovj?n G, Marton S, Klebovich I. The effect of oil as a dietary component on in vitro dissolution of an acid-labile drug. Pharmazie. 2003 Jul;58(7):502-3. PubMed PMID: 12894756. 3. Nemes KB, Abermann M, Bojti E, Gr?zal G, Al-Behaisi S, Klebovich I. Oral, intraperitoneal and intravenous pharmacokinetics of deramciclane and its N-desmethyl metabolite in the rat. J Pharm Pharmacol. 2000 Jan;52(1):47-51. PubMed PMID: 10716602. 4. Lad?nyi L, Sztruh?r I, Budai Z, Luk?cs G, Mezei T, Argay G, K?lm?n A, Simig G. Stereochemistry and enantiomeric purity of a novel anxiolytic agent, deramciclane fumarate. Chirality. 1999;11(9):689-93. PubMed PMID: 10506429.