TargetMol

Clathrodin

Product Code:
 
TAR-T27040
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27040-5mg5mg£850.00
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TAR-T27040-50mg50mg£1,661.00
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Quantity:
TAR-T27040-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
Clathrodin is a voltage-gated sodium (NaV) channels modulator.
CAS:
135383-64-1
Formula:
C11H13N5O
Molecular Weight:
231.259
Purity:
0.98
SMILES:
Nc1ncc(C=CCNC(=O)c2ccc[nH]2)[nH]1

References

1. Lillsunde KE, Toma?i? T, Kikelj D, Tammela P. Marine alkaloid oroidin analogues with antiviral potential: a novel class of synthetic compounds targeting the cellular chaperone Hsp90. Chem Biol Drug Des. 2017 Jun 5. doi: 10.1111/cbdd.13034. [Epub ahead of print] PubMed PMID: 28580714. 2. Montalv?o S, Leino TO, Kiuru PS, Lillsunde KE, Yli-Kauhaluoma J, Tammela P. Synthesis and Biological Evaluation of 2-Aminobenzothiazole and Benzimidazole Analogs Based on the Clathrodin Structure. Arch Pharm (Weinheim). 2016 Feb;349(2):137-49. doi: 10.1002/ardp.201500365. Epub 2015 Dec 28. PubMed PMID: 26709468. 3. Peigneur S, Zula A, Zidar N, Chan-Porter F, Kirby R, Madge D, Ila? J, Kikelj D, Tytgat J. Action of clathrodin and analogues on voltage-gated sodium channels. Mar Drugs. 2014 Apr 4;12(4):2132-43. doi: 10.3390/md12042132. PubMed PMID: 24714127; PubMed Central PMCID: PMC4012458. 4. Zidar N, Montalv?o S, Hodnik ?, Nawrot DA, ?ula A, Ila? J, Kikelj D, Tammela P, Ma?i? LP. Antimicrobial activity of the marine alkaloids, clathrodin and oroidin, and their synthetic analogues. Mar Drugs. 2014 Feb 14;12(2):940-63. doi: 10.3390/md12020940. PubMed PMID: 24534840; PubMed Central PMCID: PMC3944524.