TargetMol

(R)-Mequitazine

Product Code:
 
TAR-T26373
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T26373-5mg5mg£850.00
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TAR-T26373-50mg50mg£1,661.00
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Quantity:
TAR-T26373-100mg100mg£2,079.00
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Further Information

Bioactivity:
(R)-Mequitazine, a muscarinic acetylcholine receptor (M-AChRs) antagonist, is used potentially for the treatment of asthma.
CAS:
147780-50-5
Formula:
C20H22N2S
Molecular Weight:
322.47
Purity:
0.98
SMILES:
C([C@H]1CN2CCC1CC2)N1c2ccccc2Sc2ccccc12

References

1. Fonlupt P, Dubois M, Gallet H, Biot N, Pacheco H. [Changes in leukocyte phospholipid-N-methyltransferase activity after chronic treatment of allergic patients with mequitazine]. C R Seances Acad Sci III. 1983;296(21):1005-7. French. PubMed PMID: 6413002. 2. De Rotalier P, Faye M, Sissokho B, Fall D. [Allergies in ENT]. Dakar Med. 2007;52(1):2-6. French. PubMed PMID: 19102083. 3. ter Laak AM, Venhorst J, Donn?-Op den Kelder GM, Timmerman H. The histamine H1-receptor antagonist binding site. A stereoselective pharmacophoric model based upon (semi-)rigid H1-antagonists and including a known interaction site on the receptor. J Med Chem. 1995 Aug 18;38(17):3351-60. PubMed PMID: 7650688. 4. Di Bugno C, Dapporto P, Giorgi R, Manzini S, Paoli P, Subissi A, Arcamone F. Absolute configuration and biological activity of mequitamium iodide enantiomers. Chirality. 1994;6(5):382-8. PubMed PMID: 8068497.