TargetMol

Brasofensine Maleate

Product Code:
 
TAR-T26361L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

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CodeSizePrice
TAR-T26361L-5mg5mg£1,010.00
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TAR-T26361L-50mg50mg£1,982.00
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Quantity:
TAR-T26361L-100mg100mg£2,560.00
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This product comes from: United States.
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Further Information

Bioactivity:
Brasofensine Maleate inhibits the monoamine re-uptake.
CAS:
173830-14-3
Formula:
C20H24Cl2N2O5
Molecular Weight:
443.32
Purity:
0.98
SMILES:
OC(=O)C=C/C(O)=O.[H][C@]12CC[C@]([H])([C@H](C=NOC)[C@H](C1)c1ccc(Cl)c(Cl)c1)N2C

References

1. Zhu M, Whigan DB, Chang SY, Dockens RC. Disposition and metabolism of [14C]brasofensine in rats, monkeys, and humans. Drug Metab Dispos. 2008 Jan;36(1):24-35. Epub 2007 Oct 1. PubMed PMID: 17908924. 2. Minuzzi L, Olsen AK, Bender D, Arnfred S, Grant R, Danielsen EH, Cumming P. Quantitative autoradiography of ligands for dopamine receptors and transporters in brain of G?ttingen minipig: comparison with results in vivo. Synapse. 2006 Mar 15;59(4):211-9. PubMed PMID: 16385509. 3. Doudet DJ, Ruth TJ, Holden JE. Sequential versus nonsequential measurement of density and affinity of dopamine D2 receptors with [11C]raclopride: 2: effects of DAT inhibitors. J Cereb Blood Flow Metab. 2006 Jan;26(1):28-37. PubMed PMID: 15973354. 4. Johnston TH, Brotchie JM. Drugs in development for Parkinson's disease. Curr Opin Investig Drugs. 2004 Jul;5(7):720-6. Review. PubMed PMID: 15298067.