TargetMol

Rilapine

Product Code:
 
TAR-T26085
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T26085-5mg5mg£1,042.00
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TAR-T26085-50mg50mg£1,661.00
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Quantity:
TAR-T26085-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
Rilapine is an atypical antipsychotic with high affinity for the 5-HT6 receptor.
CAS:
79781-95-6
Formula:
C22H20ClN3
Molecular Weight:
361.87
Purity:
0.98
SMILES:
CN1CCN(CC1)C1=Cc2cc(Cl)ccc2C(=CC#N)c2ccccc12

References

1. Roth BL, Craigo SC, Choudhary MS, Uluer A, Monsma FJ Jr, Shen Y, Meltzer HY, Sibley DR. Binding of typical and atypical antipsychotic agents to 5-hydroxytryptamine-6 and 5-hydroxytryptamine-7 receptors. J Pharmacol Exp Ther. 1994 Mar;268(3):1403-10. PubMed PMID: 7908055. 2. Bolden C, Cusack B, Richelson E. Antagonism by antimuscarinic and neuroleptic compounds at the five cloned human muscarinic cholinergic receptors expressed in Chinese hamster ovary cells. J Pharmacol Exp Ther. 1992 Feb;260(2):576-80. PubMed PMID: 1346637. 3. Zeng XP, Le F, Richelson E. Muscarinic m4 receptor activation by some atypical antipsychotic drugs. Eur J Pharmacol. 1997 Mar 5;321(3):349-54. PubMed PMID: 9085047. 4. Roth BL, Ciaranello RD, Meltzer HY. Binding of typical and atypical antipsychotic agents to transiently expressed 5-HT1C receptors. J Pharmacol Exp Ther. 1992 Mar;260(3):1361-5. PubMed PMID: 1347569.