TargetMol

Poststatin

Product Code:
 
TAR-T25973
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T25973-5mg5mg£850.00
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Further Information

Bioactivity:
Poststatin is a prolyl endopeptidase inhibitor produced by Streptomyces viridochromogenes MH534-30F3.
CAS:
135219-43-1
Formula:
C26H48N5O7
Molecular Weight:
542.698
Purity:
0.98
SMILES:
CCC(N)CC(=O)N(C(=O)[C@@H](NC(=O)[C@@H](N)C(C)C)C(C)C)[C](=O)(CC(C)C)C(=O)N[C@@H](C(C)C)C(O)=O

References

1. Tsuda M, Muraoka Y, Someno T, Nagai M, Aoyagi T, Takeuchi T. Poststatin, a new inhibitor of prolyl endopeptidase. VI. Endopeptidase inhibitory activity of poststatin analogues containing pyrrolidine ring. J Antibiot (Tokyo). 1996 Sep;49(9):900-8. PubMed PMID: 8931724. 2. Tsuda M, Muraoka Y, Nagai M, Takeuchi T, Aoyagi T. Poststatin, a new inhibitor of prolyl endopeptidase. IV. The chemical synthesis of poststain. J Antibiot (Tokyo). 1996 Mar;49(3):287-91. PubMed PMID: 8626246. 3. Tsuda M, Muraoka Y, Nagai M, Aoyagi T, Takeuchi T. Poststatin, a new inhibitor of prolyl endopeptidase. VII. N-cycloalkylamide analogues. J Antibiot (Tokyo). 1996 Sep;49(9):909-20. PubMed PMID: 8931725. 4. Katori M, Majima M. Renal (tissue) kallikrein-kinin system in the kidney and novel potential drugs for salt-sensitive hypertension. Prog Drug Res. 2014;69:59-109. Review. PubMed PMID: 25130040.