TargetMol

Phelorphan

Product Code:
 
TAR-T25941
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T25941-5mg5mg£850.00
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TAR-T25941-50mg50mg£1,661.00
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Quantity:
TAR-T25941-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
Phelorphan is an inhibitor of enkephalinase.
CAS:
110871-16-4
Formula:
C20H22N2O4S
Molecular Weight:
386.47
Purity:
0.98
SMILES:
OC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)CS

References

1. Van Amsterdam JG, Llorens-Cortes C. Inhibition of enkephalin degradation by phelorphan: effects on striatal [Met5]enkephalin levels and jump latency in mouse hot plate test. Eur J Pharmacol. 1988 Sep 23;154(3):319-24. PubMed PMID: 3234484. 2. Haffmans J, Walsum MV, van Amsterdam JC, Dzoljic MR. Phelorphan, an inhibitor of enzymes involved in the biodegradation of enkephalins, affected the withdrawal symptoms in chronic morphine-dependent rats. Neuroscience. 1987 Jul;22(1):233-6. PubMed PMID: 2888045. 3. van Amsterdam JG, van Buuren KJ, Krielaart MJ, Zuiderveld OP, Tijms RP. Effect of inhibitors of enkephalin degradation in the isolated guinea-pig ileum. Life Sci. 1988;43(19):1529-36. PubMed PMID: 3193845. 4. Dzoljic MR. Enkephalinase inhibitors attenuate naloxone-precipitated withdrawal syndrome. NIDA Res Monogr. 1986;75:575-8. PubMed PMID: 3123978.