TargetMol

Gea 857

Product Code:
 
TAR-T25446
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T25446-5mg5mg£850.00
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TAR-T25446-50mg50mg£1,661.00
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Quantity:
TAR-T25446-100mg100mg£2,079.00
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Further Information

Bioactivity:
Gea 857 is a potassium conductance putative blocker.
CAS:
120493-42-7
Formula:
C15H22ClNO2
Molecular Weight:
283.8
Purity:
0.98
SMILES:
CC(C)[C@H](N)C(=O)OC(C)(C)Cc1ccc(Cl)cc1

References

1. Hu PS, Ross SB. NMDA receptor-mediated increase in cyclic GMP in the rat cerebellum in vivo is blocked by alaproclate and GEA-857. Pharmacol Toxicol. 1997 Feb;80(2):97-102. PubMed PMID: 9060041. 2. Ogren SO, Bartfai T, Hedlund B, Lindberg UH. GEA 857, a putative blocker of potassium conductance, enhances muscarinic agonist-evoked responses: dissociation from an action on 5-HT mechanisms. Pharmacol Toxicol. 1992 Aug;71(2):112-9. PubMed PMID: 1438027. 3. Hedlund B, Ogren SO. GEA 857 blocks potassium channels in the membrane and, thereby, prolongs muscarinic cholinergic responses in N1E-115 neuroblastoma cells. Pharmacol Toxicol. 1992 Aug;71(2):107-11. PubMed PMID: 1301072.