TargetMol

Deltakephalin

Product Code:
 
TAR-T25302
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T25302-5mg5mg£1,091.00
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TAR-T25302-50mg50mg£2,143.00
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Quantity:
TAR-T25302-100mg100mg£2,801.00
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This product comes from: United States.
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Further Information

Bioactivity:
Deltakephalin is a synthetic, potent specific opiate delta receptors agonist.
CAS:
85286-38-0
Formula:
C34H48N6O10
Molecular Weight:
700.79
Purity:
0.98
SMILES:
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@H](NC(=O)[C@@H](N)Cc1ccc(O)cc1)[C@H](C)O)C(=O)N[C@@H]([C@@H](C)O)C(O)=O

References

1. Zajac JM, Gacel G, Petit F, Dodey P, Rossignol P, Roques BP. Deltakephalin, Tyr-D-Thr-Gly-Phe-Leu-Thr: a new highly potent and fully specific agonist for opiate delta-receptors. Biochem Biophys Res Commun. 1983 Mar 16;111(2):390-7. PubMed PMID: 6301470. 2. Widy-Tyszkiewicz E, Cz?onkowski A. Analgesic activity of morphiceptin, beta-casomorphin-4, and deltakephalin in normotensive Wistar-Glaxo and spontaneously hypertensive rats. Peptides. 1989 May-Jun;10(3):539-44. PubMed PMID: 2780414. 3. Flippen-Anderson JL, Deschamps JR, Ward KB, George C, Houghten R. Crystal structure of deltakephalin: a delta-selective opioid peptide with a novel beta-bend-like conformation. Int J Pept Protein Res. 1994 Aug;44(2):97-104. PubMed PMID: 7982763. 4. Chaillet P, Coulaud A, Fourni?-Zaluski MC, Gacel G, Roques BP, Costentin J. Pain control by endogenous enkephalins is mediated by mu opioid receptors. Life Sci. 1983;33 Suppl 1:685-8. PubMed PMID: 6319920.