TargetMol

EHop-016

Product Code:
 
TAR-T2427
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T2427-5mg5mg£103.00
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TAR-T2427-1mL1 mL * 10 mM (in DMSO)£106.00
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TAR-T2427-10mg10mg£124.00
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TAR-T2427-25mg25mg£174.00
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TAR-T2427-50mg50mg£251.00
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TAR-T2427-100mg100mg£389.00
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TAR-T2427-200mg200mg£538.00
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TAR-T2427-500mg500mg£804.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
EHop-016 is a specific Rac GTPase inhibitor with IC50 of 1.1 μM for Rac1 in MDA-MB-231 and MDA-MB-435 cells, equally effective inhibition for Rac3.
CAS:
1380432-32-5
Formula:
C25H30N6O
Molecular Weight:
430.556
Pathway:
GPCR/G Protein; Cell Cycle/Checkpoint; MAPK
Purity:
0.9769
SMILES:
CCn1c2ccccc2c2cc(Nc3ccnc(NCCCN4CCOCC4)n3)ccc12
Target:
Rho; Ras

References

1. Montalvo-Ortiz BL, et al. J Biol Chem. 2012, 287(16), 13228-13238. 2. Martin H, et al. J Clin Invest. 2013, 123(10), 4449-4463.