TargetMol

K-8012

Product Code:
 
TAR-T24240
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T24240-1mg1mg£227.00
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TAR-T24240-5mg5mg£430.00
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TAR-T24240-1mL1 mL * 10 mM (in DMSO)£447.00
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TAR-T24240-10mg10mg£600.00
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TAR-T24240-25mg25mg£863.00
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Quantity:
TAR-T24240-50mg50mg£1,179.00
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Quantity:
TAR-T24240-100mg100mg£1,589.00
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Quantity:
TAR-T24240-500mg500mg£3,115.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
K-8012 is an inhibitor of the N-terminally truncated RXR.
CAS:
1346513-17-4
Formula:
C23H23FN4
Molecular Weight:
374.463
Pathway:
Metabolism
Purity:
0.98
SMILES:
CC(C)c1ccc(C=C2C(C)=C(CCc3nnn[nH]3)c3cc(F)ccc23)cc1
Target:
RAR/RXR?|Retinoid Receptor

References

1. Chen L, Wang ZG, Aleshin AE, Chen F, Chen J, Jiang F, Alitongbieke G, Zeng Z, Ma Y, Huang M, Zhou H, Cadwell G, Zheng JF, Huang PQ, Liddington RC, Zhang XK, Su Y. Sulindac-derived RXR? modulators inhibit cancer cell growth by binding to a novel site. Chem Biol. 2014 May 22;21(5):596-607. doi: 10.1016/j.chembiol.2014.02.017. Epub 2014 Apr 3. PubMed PMID: 24704507; PubMed Central PMCID: PMC4035439.