TargetMol

HTH-01-091

Product Code:
 
TAR-T24152
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T24152-1mg1mg£352.00
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Quantity:
TAR-T24152-1mL1 mL * 10 mM (in DMSO)£732.00
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Quantity:
TAR-T24152-5mg5mg£736.00
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Quantity:
TAR-T24152-10mg10mg£978.00
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Quantity:
TAR-T24152-25mg25mg£1,348.00
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Quantity:
TAR-T24152-50mg50mg£1,661.00
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Quantity:
TAR-T24152-100mg100mg£2,079.00
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Quantity:
TAR-T24152-500mg500mg£4,006.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
HTH-01-091 is a selective inhibitor of maternal embryonic leucine zipper kinase.
CAS:
2000209-42-5
Formula:
C26H28Cl2N4O2
Molecular Weight:
499.44
Pathway:
Chromatin/Epigenetic|NF-κb|JAK/STAT signaling|Metabolism|PI3K/Akt/mTOR signaling|Cell Cycle/Checkpoint|Apoptosis|Tyrosine Kinase/Adaptors
Purity:
0.98
SMILES:
CN(C)C[C@H]1CC[C@@H](CC1)N1C(=O)NCc2cnc3ccc(cc3c12)-c1cc(Cl)c(O)c(Cl)c1
Target:
Serine/threonin kinase|MELK|DYRK|Pim|RIP kinase|CDK

References

1. Huang HT, Seo HS, Zhang T, Wang Y, Jiang B, Li Q, Buckley DL, Nabet B, Roberts JM, Paulk J, Dastjerdi S, Winter GE, McLauchlan H, Moran J, Bradner JE, Eck MJ, Dhe-Paganon S, Zhao JJ, Gray NS. MELK is not necessary for the proliferation of basal-like breast cancer cells. Elife. 2017 Sep 19;6. pii: e26693. doi: 10.7554/eLife.26693. PubMed PMID: 28926338; PubMed Central PMCID: PMC5605198.