TargetMol

COR628

Product Code:
 
TAR-T23908
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T23908-5mg5mg£850.00
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TAR-T23908-50mg50mg£1,661.00
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Quantity:
TAR-T23908-100mg100mg£2,079.00
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  • Further Information
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Further Information

Bioactivity:
COR628 is the GABA(B) receptor positive allosteric modulator.
CAS:
550310-04-8
Formula:
C16H23NO3S
Molecular Weight:
309.42
Purity:
0.98
SMILES:
CCc1c(C)sc(NC(=O)C2CCCCC2)c1C(=O)OC

References

1. Mugnaini C, Pedani V, Casu A, Lobina C, Casti A, Maccioni P, Porcu A, Giunta D, Lamponi S, Solinas M, Dragoni S, Valoti M, Colombo G, Castelli MP, Gessa GL, Corelli F. Synthesis and pharmacological characterization of 2-(acylamino)thiophene derivatives as metabolically stable, orally effective, positive allosteric modulators of the GABAB receptor. J Med Chem. 2013 May 9;56(9):3620-35. doi: 10.1021/jm400144w. Epub 2013 Apr 18. PubMed PMID: 23544432. 2. Castelli MP, Casu A, Casti P, Lobina C, Carai MA, Colombo G, Solinas M, Giunta D, Mugnaini C, Pasquini S, Tafi A, Brogi S, Gessa GL, Corelli F. Characterization of COR627 and COR628, two novel positive allosteric modulators of the GABA(B) receptor. J Pharmacol Exp Ther. 2012 Mar;340(3):529-38. doi: 10.1124/jpet.111.186460. Epub 2011 Nov 30. PubMed PMID: 22129594.