TargetMol

CAY10499

Product Code:
 
TAR-T22637
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T22637-5mg5mg£164.00
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Quantity:
TAR-T22637-10mg10mg£234.00
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TAR-T22637-25mg25mg£428.00
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This product comes from: United States.
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Further Information

Bioactivity:
CAY10499 is a potent inhibitor of monoglyceride lipase (MGL) and human hormone-sensitive lipase. CAY10499 inhibited MGL-mediated 4-NPA hydrolysis with the IC 50 value of 0.5 ? 0.03 μM. CAY10499 fully inhibited [3H]-AEA hydrolysis by human recombinant FAAH with an IC50 of 76 nM. CAY10499 displaced only 25% and 20% of [3H]-CP-55940-specific binding to the CB1 and CB2 receptors, respectively [1]. CAY10499 potently inhibited the activity of human hormone-sensitive lipase with an IC50 of 90 nM for the recombinant human hormone-sensitive lipase enzyme [1][2].
CAS:
T22637
Formula:
C18H17N3O5
Molecular Weight:
355.3
Purity:
0.98
SMILES:
CC1=CC(N(N=C(O2)OC)C2=O)=CC=C1NC(OCC3=CC=CC=C3)=O