TargetMol

PF-02575799

Product Code:
 
TAR-T16158
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T16158-5mg5mg£1,010.00
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TAR-T16158-50mg50mg£1,982.00
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Quantity:
TAR-T16158-100mg100mg£2,560.00
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This product comes from: United States.
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Further Information

Bioactivity:
PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77?0.29 nM).
CAS:
863491-70-7
Formula:
C42H37FN4O4
Molecular Weight:
680.78
Pathway:
Neuroscience; GPCR/G Protein
Purity:
0.98
SMILES:
CC(C)Oc1ccc(cc1)-c1ccccc1C(=O)Nc1ccc2cc(ccc2n1)C(=O)N[C@H](C(=O)N(C)Cc1ccc(F)cc1)c1ccccc1
Target:
Adenosine Receptor

References

1. Robinson RP, et al. Discovery of microsomal triglyceride transfer protein (MTP) inhibitors with potential for decreased active metabolite load compared to dirlotapide. Bioorg Med Chem Lett. 2011 Jul 15;21(14):4150-4.