TargetMol

EML 425

Product Code:
 
TAR-T15216
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15216-1mg1mg£101.00
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TAR-T15216-5mg5mg£142.00
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TAR-T15216-1mL1 mL * 10 mM (in DMSO)£149.00
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TAR-T15216-10mg10mg£195.00
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TAR-T15216-25mg25mg£340.00
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TAR-T15216-50mg50mg£475.00
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TAR-T15216-100mg100mg£658.00
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This product comes from: United States.
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Further Information

Bioactivity:
EML 425 is a potent and selective inhibitor of CREB binding protein (CBP)/p300 (IC50s: 2.9 and 1.1 μM, respectively).
CAS:
1675821-32-5
Formula:
C27H24N2O4
Molecular Weight:
440.499
Pathway:
Chromatin/Epigenetic
Purity:
1
SMILES:
Cc1cc(O)cc(C)c1C=C1C(=O)N(Cc2ccccc2)C(=O)N(Cc2ccccc2)C1=O
Target:
Epigenetic Reader Domain; Histone Acetyltransferase

References

1. Milite C, et al. A novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach. J Med Chem. 2015 Mar 26;58(6):2779-98.