TargetMol

EBI-1051

Product Code:
 
TAR-T15193
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

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CodeSizePrice
TAR-T15193-5mg5mg£1,332.00
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TAR-T15193-50mg50mg£2,625.00
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Quantity:
TAR-T15193-100mg100mg£3,524.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
EBI-1051 is a highly potent and orally efficacious inhibitor of MEK (IC50: 3.9 nM).
CAS:
1801896-05-8
Formula:
C18H15F2IN2O5
Molecular Weight:
504.228
Pathway:
MAPK
Purity:
0.98
SMILES:
OCC(CO)ONC(=O)c1cc2ccoc2c(F)c1Nc1ccc(I)cc1F
Target:
MEK

References

1. Lu B, et al. Discovery of EBI-1051: A novel and orally efficacious MEK inhibitor with benzofuran scaffold. Bioorg Med Chem. 2018 Feb 1;26(3):581-589.