TargetMol

Draflazine

Product Code:
 
TAR-T15167
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15167-5mg5mg£850.00
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TAR-T15167-50mg50mg£1,661.00
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Quantity:
TAR-T15167-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
Draflazine is an ENT1 inhibitor. It completely reverses the hypersensitivity in the complete Freund?s adjuvant (CFA) model of mechanical hyperalgesia. Draflazine also completely reverses the hypersensitivity of the carrageenan inflammation model of thermal and mechanical hyperalgesia.
CAS:
120770-34-5
Formula:
C30H33Cl2F2N5O2
Molecular Weight:
604.52
Purity:
0.98
SMILES:
NC(=O)C1CN(CCCCC(c2ccc(F)cc2)c2ccc(F)cc2)CCN1CC(=O)Nc1c(Cl)cc(N)cc1Cl

References

1. Maes SS, et al. Antihyperalgesic activity of nucleoside transport inhibitors in models of inflammatory pain in guinea pigs. J Pain Res. 2012;5:391-400.