TargetMol

BMS-986163

Product Code:
 
TAR-T14686
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T14686-5mg5mg£1,332.00
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TAR-T14686-50mg50mg£2,625.00
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Quantity:
TAR-T14686-100mg100mg£3,524.00
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This product comes from: United States.
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Further Information

Bioactivity:
BMS-986163 is a negative allosteric modulator of GluN2B and the prodrug BMS-986163 rapidly converts to its active parent molecule BMS-986169 (Ki=4 nM, IC50=24 nM).
CAS:
1801151-09-6
Formula:
C23H28FN2O5P
Molecular Weight:
462.458
Purity:
0.98
SMILES:
Cc1ccc(CN2CC[C@@H](N3CC[C@H]([C@H](F)C3)c3ccc(OP(O)(O)=O)cc3)C2=O)cc1

References

1. Marcin LR, et al. BMS-986163, a Negative Allosteric Modulator of GluN2B with Potential Utility in Major Depressive Disorder. ACS Med Chem Lett. 2018 Apr 13;9(5):472-477.