TargetMol

BAY-299

Product Code:
 
TAR-T14502
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T14502-5mg5mg£105.00
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Quantity:
TAR-T14502-1mL1 mL * 10 mM (in DMSO)£109.00
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Quantity:
TAR-T14502-10mg10mg£127.00
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TAR-T14502-25mg25mg£185.00
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Quantity:
TAR-T14502-50mg50mg£274.00
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Quantity:
TAR-T14502-100mg100mg£429.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
BAY-299 is an effecitve inhibitor of the bromodomain and PHD finger family member BRPF2 and the TATA box binding protein-associated factors TAF1 and TAF1L with IC50s of 67 nM, 8 nM, and 106 nM, respectively.
CAS:
2080306-23-4
Formula:
C25H23N3O4
Molecular Weight:
429.47
Pathway:
Proteases/Proteasome; Chromatin/Epigenetic
Purity:
0.975
SMILES:
Cc1cc2n(C)c(=O)n(C)c2cc1N1C(=O)c2cccc3c(CCCO)ccc(C1=O)c23
Target:
Epigenetic Reader Domain; Carboxypeptidase

References

1. Bouch? L, et al. Benzoisoquinolinediones as Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains. J Med Chem. 2017 May 11;60(9):4002-4022.