TargetMol

SNT-207858

Product Code:
 
TAR-T12946
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12946-5mg5mg£850.00
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Quantity:
TAR-T12946-50mg50mg£1,661.00
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Quantity:
TAR-T12946-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
SNT-207858 is a selective, blood brain barrier penetrating, potent and orally active antagonist of melanocortin-4 (MC-4) receptor. SNT207858 has an IC50 of 22 nM (binding) and 11 nM (function) on the MC-4 receptor.
CAS:
1104080-42-3
Formula:
C32H45Cl4N5O3
Molecular Weight:
689.54
Purity:
0.98
SMILES:
Cl.Cl.CC[C@H](COc1cccnc1C1CCN(CC1)C(=O)[C@@H](Cc1ccc(Cl)cc1Cl)NC(=O)N1CCCC1)N1CCCC1

References

1. Weyermann P, et al. Orally available selective melanocortin-4 receptor antagonists stimulate food intake and reduce cancer-induced cachexia in mice. PLoS One. 2009;4(3):e4774.