TargetMol

RP-001 hydrochloride

Product Code:
 
TAR-T12780L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12780L-5mg5mg£1,171.00
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TAR-T12780L-50mg50mg£2,303.00
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Quantity:
TAR-T12780L-100mg100mg£3,042.00
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This product comes from: United States.
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Further Information

Bioactivity:
RP-001 hydrochloride is a selective agonist of picomolar short-acting S1P1 (EDG1)(EC50 of 9 pM), has little activity on S1P2-S1P4 and only moderate affinity for S1P5.
CAS:
1781880-34-9
Formula:
C24H25ClN4O4
Molecular Weight:
468.94
Purity:
0.98
SMILES:
Cl.CC(C)Oc1ccc(cc1C#N)-c1nc(no1)-c1cccc2C(CCc12)NCCC(O)=O

References

1. Cahalan SM, et al. Actions of a picomolar short-acting S1P? agonist in S1P?-eGFP knock-in mice. Nat Chem Biol. 2011 May;7(5):254-6.