TargetMol

Astemizole

Product Code:
 
TAR-T1278
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T1278-5mg5mg£104.00
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Quantity:
TAR-T1278-1mL1 mL * 10 mM (in DMSO)£107.00
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TAR-T1278-10mg10mg£117.00
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Quantity:
TAR-T1278-25mg25mg£146.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Astemizole is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 receptors, with less anticholinergic effects compared to related agents. It is a long-acting, non-sedative antihistaminic used in the treatment of seasonal allergic rhinitis, asthma, allergic conjunctivitis, and chronic idiopathic urticaria.
CAS:
68844-77-9
Formula:
C28H31FN4O
Molecular Weight:
458.581
Pathway:
Membrane transporter/Ion channel; Immunology/Inflammation; GPCR/G Protein; Neuroscience
Purity:
0.9988
SMILES:
COc1ccc(CCN2CCC(CC2)Nc2nc3ccccc3n2Cc2ccc(F)cc2)cc1
Target:
Potassium Channel; Histamine Receptor

References

1. Salata JJ, et al. Circ Res. 1995 Jan;76(1):110-9.