TargetMol

Rivanicline

Product Code:
 
TAR-T12738L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12738L-5mg5mg£850.00
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TAR-T12738L-50mg50mg£1,661.00
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Quantity:
TAR-T12738L-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
Rivanicline is a neuronal nicotinic receptor agonist, showing high selectivity for the α4β2 subtype (Ki=26 nM). It show > 1,000 fold selectivity than α7 receptors(Ki= 36000 nM and IC50 : 26 nM).
CAS:
15585-43-0
Formula:
C10H14N2
Molecular Weight:
162.236
Purity:
0.98
SMILES:
CNCCC=Cc1cccnc1

References

1. Bencherif M, et al. RJR-2403: a nicotinic agonist with CNS selectivity I. In vitro characterization. J Pharmacol Exp Ther. 1996 Dec;279(3):1413-21. 2. Lippiello PM, et al. RJR-2403: a nicotinic agonist with CNS selectivity II. In vivo characterization. J Pharmacol Exp Ther. 1996 Dec;279(3):1422-9. 3. Damaj MI, et al. Antinociceptive and pharmacological effects of metanicotine, a selective nicotinic agonist. J Pharmacol Exp Ther. 1999 Oct;291(1):390-8.