TargetMol

OTS186935 trihydrochloride

Product Code:
 
TAR-T12344L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T12344L-5mg5mg£850.00
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TAR-T12344L-50mg50mg£1,661.00
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Quantity:
TAR-T12344L-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
OTS186935 trihydrochloride is a protein methyltransferase inhibitor of SUV39H2(IC50 of 6.49 nM).
CAS:
2093401-85-3
Formula:
C25H29Cl4N5O2
Molecular Weight:
573.34
Purity:
0.98
SMILES:
Cl.Cl.Cl.COc1cc(OC)c(cc1Cl)-c1cn2ccc(cc2n1)N1CC[C@@H](C1)NCc1ccncc1

References

1. Vougiouklakis T, et al. Development of novel SUV39H2 inhibitors that exhibit growth suppressive effects in mouse xenograft models and regulate the phosphorylation of H2AX. Oncotarget. 2018 Aug 7;9(61):31820-31831.