TargetMol

MT-3014

Product Code:
 
TAR-T12119
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12119-5mg5mg£1,010.00
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TAR-T12119-50mg50mg£1,982.00
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Quantity:
TAR-T12119-100mg100mg£2,560.00
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This product comes from: United States.
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Further Information

Bioactivity:
MT-3014 is a potent, highly selective and brain-penetrated inhibitor of phosphodiesterase 10A (PDE 10A)(human PDE 10A and bovine PDE 10A with IC50s of 0.062 nM and 0.09 nM , respectively).
CAS:
1332727-40-8
Formula:
C23H25F2N7O
Molecular Weight:
453.498
Purity:
0.98
SMILES:
Cc1nc2ccc(F)cc2nc1-c1cc2nc(cc(NCC(C)(C)O)n2n1)N1CC[C@@H](F)C1

References

1. Koizumi Y, et al. Discovery of a pyrazolo[1,5-a]pyrimidine derivative (MT-3014) as a highly selective PDE10A inhibitor via core structure transformation from the stilbene moiety. Bioorg Med Chem. 2019 Jun 19.