TargetMol

L-45 dihydrochloride (2079885-05-3 free base)

Product Code:
 
TAR-T11796
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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TAR-T11796-100mg100mgEnquire
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TAR-T11796-5mg5mg£243.00
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TAR-T11796-10mg10mg£384.00
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Further Information

Bioactivity:
L-45 dihydrochloride is the first selective, potent, and cell-active p300/CBP-associated factor (PCAF) bromodomain (Brd) inhibitor with a Kd of 126?15 nM.
CAS:
T11796
Formula:
C21H26Cl2N6
Molecular Weight:
433.38
Purity:
0.98
SMILES:
C[C@@H]([C@H](C1=CC=CC=C1)N(C)C)NC(C2=C3C=CC=C2)=NN4C3=NN=C4C.[H]Cl.[H]Cl

References

1. Moustakim M, et al. Discovery of a PCAF Bromodomain Chemical Probe. Angew Chem Int Ed Engl. 2017 Jan 16;56(3):827-831.