TargetMol

GSK1521498 free base

Product Code:
 
TAR-T11478L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T11478L-5mg5mg£304.00
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Quantity:
TAR-T11478L-50mg50mg£1,396.00
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Quantity:
TAR-T11478L-100mg100mg£2,079.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GSK1521498 free base is a potent and selective antagonist of the μ-opioid receptor. GSK1521498 free base also has the potential for disorders of compulsive consumption of food, alcohol, and drugs.
CAS:
1007573-18-3
Formula:
C24H20F2N4
Molecular Weight:
402.449
Pathway:
Endocrinology/Hormones; Neuroscience; GPCR/G Protein
Purity:
0.98
SMILES:
Fc1cc(cc(F)c1CNC1Cc2ccccc2C1)-c1cccc(c1)-c1ncn[nH]1
Target:
Opioid Receptor

References

1. Giuliano C, et al. The Novel ?-Opioid Receptor Antagonist GSK1521498 Decreases Both Alcohol Seeking and Drinking: Evidence from a New Preclinical Model of Alcohol Seeking. Neuropsychopharmacology. 2015 Dec;40(13):2981-92.