TargetMol

GSK 366

Product Code:
 
TAR-T11470
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11470-5mg5mg£724.00
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TAR-T11470-50mg50mg£2,625.00
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Quantity:
TAR-T11470-100mg100mg£3,524.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GSK 366 is a potent kynurenine-3-monooxygenase (KMO) inhibitor (IC50s: 0.7 nM and 2.3 nM for P. fluorescens-KMO and human KMO).
CAS:
1953157-39-5
Formula:
C17H16ClN3O4
Molecular Weight:
361.78
Pathway:
Metabolism
Purity:
0.98
SMILES:
C[C@@H](Oc1cc2onc(CCC(O)=O)c2cc1Cl)c1ccc(C)nn1
Target:
Hydroxylase

References

1. Hutchinson JP, et al. Structural and mechanistic basis of differentiated inhibitors of the acute pancreatitis target kynurenine-3-monooxygenase. Nat Commun. 2017 Jun 12;8:15827.