TargetMol

FAK inhibitor 2

Product Code:
 
TAR-T11260
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11260-5mg5mg£304.00
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TAR-T11260-50mg50mg£1,364.00
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Quantity:
TAR-T11260-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
FAK inhibitor 2, antitumor and anti-angiogenesis activitiesis ,is a potent focal adhesion kinase (FAK) inhibitor with an IC50 of 0.07 nM .
CAS:
2354405-14-2
Formula:
C29H33F3N8O2S2
Molecular Weight:
646.75
Pathway:
Cytoskeletal Signaling; Tyrosine Kinase/Adaptors; Angiogenesis
Purity:
0.98
SMILES:
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N2CCN(CC2)C(=S)SCCN(C)C)ncc1C(F)(F)F
Target:
FAK

References

1. Su Y, et al. Discovery of 2,4-diarylaminopyrimidine derivatives bearing dithiocarbamate moiety as novel FAK inhibitors with antitumor and anti-angiogenesis activities. Eur J Med Chem. 2019 May 18;177:32-46.