TargetMol

ERK2 IN-1

Product Code:
 
TAR-T11228
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11228-5mg5mg£1,251.00
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Quantity:
TAR-T11228-50mg50mg£2,464.00
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Quantity:
TAR-T11228-100mg100mg£3,283.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
ERK2 IN-1 is a selective ERK2 inhibitor with an IC50 of 7 nM.
CAS:
1093061-47-2
Formula:
C36H34FN7O2S
Molecular Weight:
647.77
Pathway:
MAPK
Purity:
0.98
SMILES:
CS[C@]1(CCN(CC(=O)N2CCC(=CC2)c2ccc(cc2)-c2ncccn2)C1)C(=O)Nc1ccc2[nH]nc(-c3ccc(F)cc3)c2c1
Target:
ERK

References

1. Boga SB, Discovery of 3(S)-thiomethyl pyrrolidine ERK inhibitors for oncology. Bioorg Med Chem Lett. 2018 Jun 15;28(11):2029-2034.