TargetMol

DRAK2-IN-1

Product Code:
 
TAR-T11094
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11094-5mg5mg£244.00
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TAR-T11094-50mg50mg£870.00
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Quantity:
TAR-T11094-100mg100mg£1,468.00
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This product comes from: United States.
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Further Information

Bioactivity:
Drak2-in-1, a potent, selective and ATP-competitive DRAK2 inhibitor, has an IC50 and KIvalue of 3 nM and 0.26 nM, respectively.Drak2-in-1 also had an effect on DRAK1 (IC50=51 nM).
CAS:
871837-60-4
Formula:
C21H20N4O3
Molecular Weight:
376.416
Purity:
0.98
SMILES:
CCCCC(=O)Nc1ccc2NC(=O)C(=C3/Nc4ccccc4/C/3=N/O)c2c1

References

1. Jung ME, et al.Discovery of indirubin derivatives as new class of DRAK2 inhibitors from high throughput screening.Bioorg Med Chem Lett.?2016 Jun 1;26(11):2719-23