TargetMol

AHR antagonist 4

Product Code:
 
TAR-T10271
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10271-5mg5mg£1,091.00
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TAR-T10271-50mg50mg£2,143.00
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Quantity:
TAR-T10271-100mg100mg£2,801.00
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This product comes from: United States.
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Further Information

Bioactivity:
AHR antagonist 4 is a potent aryl hydrocarbon receptor (AHR) antagonist extracted from patent WO2018146010A1 (example 293; IC50: 82.2 nM). It has anti-cancer effects.
CAS:
2242465-58-1
Formula:
C20H14F6N4O4
Molecular Weight:
488.346
Purity:
0.98
SMILES:
O[C@@H](CNC(=O)c1cc(nn(-c2cccnc2)c1=O)-c1ccc(OC(F)(F)F)cc1)C(F)(F)F

References

1. Ilona GUTCHER, et al. 2-heteroaryl-3-oxo-2,3-dihydropyridazine-4-carboxamides for the treatment of cancer. WO2018146010A1.