TargetMol

ASP2905

Product Code:
 
TAR-T9070
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T9070-1mg1mg£95.00
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TAR-T9070-2mg2mg£103.00
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TAR-T9070-5mg5mg£122.00
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TAR-T9070-1mL1 mL * 10 mM (in DMSO)£127.00
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TAR-T9070-10mg10mg£148.00
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TAR-T9070-25mg25mg£230.00
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TAR-T9070-50mg50mg£334.00
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TAR-T9070-100mg100mg£503.00
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Further Information

Bioactivity:
ASP-2905 is a potent and selective?inhibitor of potassium channel Kv12.2 encoded by the Kcnh3/BEC1 gene. It can cross the blood-brain barrier and has antipsychotic activities
CAS:
792184-90-8
Formula:
C20H17FN8
Molecular Weight:
388.41
Pathway:
Membrane transporter/Ion channel
Purity:
0.9829
SMILES:
Fc1ccc(Nc2nc(NCc3ncccn3)nc(Nc3ccccc3)n2)cc1
Target:
Potassium Channel

References

Shinji Takahashi, et al. Neurochemical and neuropharmacological characterization of ASP2905, a novel potent selective inhibitor of the potassium channel KCNH3. Eur J Pharmacol. 2017 Sep 5;810:26-35. Shinji Takahashi, et al. ASP2905, a specific inhibitor of the potassium channel Kv12.2 encoded by the Kcnh3 gene, is psychoactive in mice. Behav Brain Res. 2020 Jan 27;378:112315.