TargetMol

EN4

Product Code:
 
TAR-T9061
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T9061-1mg1mg£96.00
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TAR-T9061-5mg5mg£128.00
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TAR-T9061-1mL1 mL * 10 mM (in DMSO)£134.00
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TAR-T9061-10mg10mg£142.00
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TAR-T9061-25mg25mg£229.00
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TAR-T9061-50mg50mg£309.00
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Quantity:
TAR-T9061-100mg100mg£430.00
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Further Information

Bioactivity:
EN4 MYC inhibitor is a covalent ligand that targets cysteine 171 (C171) of MYC. It is selective for c-MYC over N-MYC and L-MYC, and inhibits MYC transcriptional activity, downregulates MYC targets, and impairs tumorigenesis.
CAS:
1197824-15-9
Formula:
C25H24N2O4
Molecular Weight:
416.477
Pathway:
Cell Cycle/Checkpoint
Purity:
0.9819
SMILES:
CCOc1ccc(Oc2ccccc2NC(=O)c2ccc(CNC(=O)C=C)cc2)cc1
Target:
c-Myc

References

Lydia Boike, et al. Discovery of a Functional Covalent Ligand Targeting an Intrinsically Disordered Cysteine within MYC. Cell Chem Biol. 2021 Jan 21;28(1):4-13.e17.