TargetMol

ML382

Product Code:
 
TAR-T8538
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T8538-1mg1mg£95.00
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TAR-T8538-5mg5mg£125.00
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TAR-T8538-1mL1 mL * 10 mM (in DMSO)£132.00
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TAR-T8538-10mg10mg£161.00
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TAR-T8538-25mg25mg£246.00
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TAR-T8538-50mg50mg£389.00
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TAR-T8538-100mg100mg£544.00
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This product comes from: United States.
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Further Information

Bioactivity:
ML382 is a potent and selective MrgX1 positive allosteric modulator(EC50 : 190 nM).
CAS:
1646499-97-9
Formula:
C18H20N2O4S
Molecular Weight:
360.43
Purity:
0.9971
SMILES:
CCOc1ccccc1NC(=O)c1ccccc1NS(=O)(=O)C1CC1

References

Li Z, et al. Targeting human Mas-related G protein-coupled receptor X1 to inhibit persistent pain. Proc Natl Acad Sci U S A. 2017;114(10):E1996-E2005. Wen W, et al. Discovery and characterization of 2-(cyclopropanesulfonamido)-N-(2-ethoxyphenyl)benzamide, ML382: a potent and selective positive allosteric modulator of MrgX1. ChemMedChem. 2015;10(1):57-61.