TargetMol

Eltoprazine hydrochloride

Product Code:
 
TAR-T7498
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
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CodeSizePrice
TAR-T7498-2mg2mg£96.00
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TAR-T7498-5mg5mg£111.00
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TAR-T7498-1mL1 mL * 10 mM (in DMSO)£116.00
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TAR-T7498-10mg10mg£142.00
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TAR-T7498-25mg25mg£213.00
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TAR-T7498-50mg50mg£334.00
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TAR-T7498-100mg100mg£462.00
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Further Information

Bioactivity:
Eltoprazine hydrochloride is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM, respectively).
CAS:
98206-09-8
Formula:
C12H17ClN2O2
Molecular Weight:
256.73
Pathway:
GPCR/G Protein; Neuroscience
Purity:
0.9994
SMILES:
Cl.C1CN(CCN1)c1cccc2OCCOc12
Target:
5-HT Receptor

References

Boer S F D , Lesourd M , Mocaer E , et al. Selective Antiaggressive Effects of Alnespirone in Resident-Intruder Test Are Mediated via 5-Hydroxytryptamine1A Receptors: A Comparative Pharmacological Study with 8-Hydroxy-2-Dipropylaminotetralin, Ipsapirone, Buspirone, Eltoprazine, and WAY-100635[J]. Journal of Pharmacology & Experimental Therapeutics, 1999, 288(3):1125-1133. Gravius A , Dekundy A , Vanaga A , et al. Further pharmacological characterization of eltoprazine: Focus on its anxiolytic, anorexic, and adverse-effect potential[J]. Acta neurobiologiae experimentalis, 2017, 77(1):77-85.