TargetMol

BRD9539

Product Code:
 
TAR-T7378
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7378-2mg2mg£95.00
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TAR-T7378-5mg5mg£108.00
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TAR-T7378-1mL1 mL * 10 mM (in DMSO)£112.00
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TAR-T7378-10mg10mg£134.00
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TAR-T7378-25mg25mg£177.00
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TAR-T7378-50mg50mg£227.00
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Quantity:
TAR-T7378-100mg100mg£302.00
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Further Information

Bioactivity:
BRD9539 is an inhibitor of euchromatin histone methyltransferase 2 (EHMT2), also known as G9a, with an IC50 value of 6.3 μM
CAS:
1374601-41-8
Formula:
C24H21N3O3
Molecular Weight:
399.45
Pathway:
Chromatin/Epigenetic
Purity:
0.98
SMILES:
OC(=O)c1ccc2n(CCCc3ccccc3)c(NC(=O)c3ccccc3)nc2c1
Target:
Histone Methyltransferase

References

Yuan Y , Wang Q , Paulk J , et al. A Small-Molecule Probe of the Histone Methyltransferase G9a Induces Cellular Senescence in Pancreatic Adenocarcinoma[J]. ACS Chemical Biology, 2012, 7(7):1152-1157.